SCHEMBL4707185

SCHEMBL4707185

FC(F)(F)c1cc(Cn2nnc(C3=NCCN3Cc3cccc(Cl)c3Cl)c2-c2ccccc2)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.37
MAP4K4 O95819 2/20 0.37
PIM1 P11309 2/20 0.37
PRKACA P17612 2/20 0.37
CDK2 P24941 2/20 0.37
GSK3B P49841 2/20 0.37
HIPK2 Q9H2X6 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
GRM2 Q14416 2/20 0.36
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IDO1 P14902 2/20 0.34
PLK4 O00444 1/20 0.34
AURKA O14965 1/20 0.34
MAPK13 O15264 1/20 0.34
DAPK3 O43293 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708192 0.94 SMN1; SMN2 (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4707422 0.88 SMN1; SMN2 (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4707796 0.87 CDC7 (0.39) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4707135 0.87 IDO1 (0.39) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4709645 0.80 CDC7 (0.38) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4705897 0.79 PTAFR (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4706657 0.78 ALDH1A1 (0.42) ALDH1A1HPGDSMN1; SMN2SLC16A3SLC16A1
SCHEMBL4758977 0.78 GABRA2 (0.37) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4790291 0.76 PTGER4 (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4705280 0.76 PTGER4 (0.40) CDC7MAP4K4PIM1PRKACACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed