SCHEMBL4708022

SCHEMBL4708022

O=CCc1cc(Cl)ccc1-c1nnn[nH]1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
IDO1 P14902 2/20 0.33
PPOX P50336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1196827 0.81 CYP2A6 (0.34) ALDH1A1MAPTIDO1
SCHEMBL29792715 0.81 MEN1 (0.30) MAPTIDO1
SCHEMBL23088225 0.81 MEN1 (0.30) MAPTIDO1
SCHEMBL31220830 0.81 CYP2A6 (0.34) ALDH1A1MAPTIDO1
Hydrochloric Acid SCHEMBL21355478 0.79 CYP2A6 (0.33) IDO1
SCHEMBL27033835 0.79 KEAP1 (0.40) ALDH1A1MAPT
SCHEMBL29958529 0.79 KEAP1 (0.40) ALDH1A1MAPT
SCHEMBL3633061 0.78 XDH (0.51) XDHALDH1A1MAPTIDO1PPOX
SCHEMBL2236405 0.77 FFAR1 (0.40)
SCHEMBL23088189 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS Brystol-Myers Squibb Company (US) 2008-10-22 EP disclosed
WO-2007070826-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-21 WO disclosed