SCHEMBL4708046

SCHEMBL4708046

O=C(c1ccccc1Cl)c1ccncc1-c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORB Q92753 5/20 0.42
RORC P51449 3/20 0.42
TACR1 P25103 2/20 0.39
IDH1 O75874 1/20 0.38
GPBAR1 Q8TDU6 9/20 0.38
GRM2 Q14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708172 0.94 RORB (0.46) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4707863 0.93 IDH1 (0.44) RORBRORCTACR1IDH1GPBAR1
SCHEMBL4708296 0.93 RORB (0.41) RORBRORCTACR1IDH1GPBAR1
SCHEMBL4709807 0.89 RORB (0.40) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4706972 0.89 RORB (0.40) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4705938 0.89 RORB (0.37) RORBRORCTACR1IDH1GPBAR1
SCHEMBL4708209 0.88 RORB (0.39) RORBRORCTACR1IDH1GRM2
SCHEMBL4705184 0.88 TACR1 (0.44) RORBRORCTACR1GPBAR1
SCHEMBL4757295 0.88 RORB (0.51) RORBRORCTACR1GRM2
Tradipitant SCHEMBL2898629 0.87 RORB (0.42) RORBRORCTACR1IDH1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed