SCHEMBL4707863

SCHEMBL4707863

O=C(c1ccccc1Cl)c1ccncc1-c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.44
RORB Q92753 5/20 0.43
RORC P51449 4/20 0.43
TACR1 P25103 1/20 0.38
GPBAR1 Q8TDU6 8/20 0.38
GRM2 Q14416 1/20 0.36
CRHR1 P34998 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708296 0.93 RORB (0.41) IDH1RORBRORCTACR1GPBAR1
SCHEMBL4708046 0.93 RORB (0.42) IDH1RORBRORCTACR1GPBAR1
SCHEMBL4705371 0.89 IDH1 (0.43) IDH1RORBRORCGPBAR1GRM2
SCHEMBL4706229 0.89 IDH1 (0.44) IDH1RORBRORCGPBAR1GRM2
SCHEMBL4707854 0.89 IDH1 (0.43) IDH1RORBRORCTACR1GPBAR1
SCHEMBL4706972 0.88 RORB (0.40) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4709807 0.88 RORB (0.40) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4708172 0.87 RORB (0.46) RORBRORCTACR1GPBAR1GRM2
SCHEMBL4705184 0.86 TACR1 (0.44) RORBRORCTACR1GPBAR1
SCHEMBL4707706 0.86 IDH1 (0.42) IDH1RORBRORCTACR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed