SCHEMBL4708323

SCHEMBL4708323

Nc1ccnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2cnccn2)c1C(=O)c1ccccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 9/20 0.38
RORC P51449 5/20 0.38
P2RX7 Q99572 2/20 0.33
USP2 O75604 2/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
IDH1 O75874 1/20 0.32
CYP2D6 P10635 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
TACR1 P25103 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.32
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708052 0.89 IDH1 (0.41) RORBRORCCYP3A4IDH1CYP2D6
SCHEMBL4708632 0.89 RORB (0.42) RORBRORCIDH1TACR1GABRA2
SCHEMBL4707462 0.88 RORB (0.41) RORBRORCIDH1
SCHEMBL4706074 0.88 RORB (0.39) RORBRORCP2RX7USP2MEN1
SCHEMBL4705407 0.88 RORB (0.42) RORBRORCTACR1GABRA2GABRB2
Water SCHEMBL4707272 0.88 RORB (0.41) RORBRORCTACR1GABRA2GABRB2
Water SCHEMBL4707271 0.88 RORB (0.41) RORBRORCTACR1GABRA2GABRB2
SCHEMBL4706528 0.85 RORB (0.36) RORBRORCP2RX7USP2MEN1
SCHEMBL4708328 0.85 RORB (0.41) RORBRORCHTTHSD17B10TACR1
SCHEMBL4709807 0.84 RORB (0.40) RORBRORCP2RX7TACR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed