SCHEMBL4708632

SCHEMBL4708632

Nc1ccnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2cncnc2)c1C(=O)c1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RORB Q92753 12/20 0.42
RORC P51449 5/20 0.42
IDH1 O75874 1/20 0.34
CDC7 O00311 1/20 0.33
GRM2 Q14416 1/20 0.33
TACR1 P25103 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708052 0.93 IDH1 (0.41) RORBRORCIDH1GABRA2GABRB2
SCHEMBL4707462 0.92 RORB (0.41) RORBRORCIDH1CDC7GRM2
SCHEMBL4705407 0.92 RORB (0.42) RORBRORCCDC7TACR1GABRA2
Water SCHEMBL4707272 0.91 RORB (0.41) RORBRORCCDC7TACR1GABRA2
Water SCHEMBL4707271 0.91 RORB (0.41) RORBRORCCDC7TACR1GABRA2
SCHEMBL4706766 0.91 RORB (0.43) RORBRORCIDH1CDC7GRM2
SCHEMBL4708323 0.89 RORB (0.38) RORBRORCIDH1TACR1GABRA2
SCHEMBL4705482 0.88 RORB (0.41) RORBRORCIDH1GRM2TACR1
SCHEMBL6385997 0.87 RORB (0.42) RORBRORCIDH1CDC7GRM2
SCHEMBL4708328 0.86 RORB (0.41) RORBRORCCDC7TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed