SCHEMBL4709530

SCHEMBL4709530

COc1ccc(CN2C=C3NC(NCCc4ccc(C(F)(F)F)cc4Cl)=NC(C(C(=O)O)c4cccnc4)=C3N2)cc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
DGAT2 Q96PD7 5/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
CHEK1 O14757 3/20 0.33
THRB P10828 1/20 0.33
PTGDR Q13258 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
FFAR1 O14842 1/20 0.32
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
KCNA5 P22460 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4709695 0.94 CYP3A4 (0.33) CYP3A4DGAT2LMNATP53MAPT
SCHEMBL4095980 0.84 PTGDR (0.33) CYP3A4DGAT2LMNATP53MAPT
SCHEMBL4709531 0.64 CYP3A4 (0.35) CYP3A4LMNATP53MAPTMEN1
SCHEMBL4271062 0.59 ACP1 (0.39) LMNATP53MAPTMEN1KMT2A
SCHEMBL3069012 0.56 FFAR1 (0.47) MAPTMEN1KMT2AFFAR1KCNA5
SCHEMBL11183822 0.54 CHRNB2 (0.44) CYP3A4LMNAMAPTMEN1KMT2A
SCHEMBL1581284 0.54 ACP1 (0.53) CYP3A4LMNATP53MAPTMEN1
SCHEMBL11612621 0.53 ATM (0.77) CYP3A4KMT2ACTSLCTSSKCNA5
SCHEMBL7057097 0.53 GAA (0.47) CYP3A4TP53THRBMEN1KMT2A
SCHEMBL6491361 0.53 ITGB3 (0.60) KMT2AFFAR1KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1903045-A1 PYRAZOLOPYRIMIDINE DERIVATIVE Mitsubishi Tanabe Pharma Corporation (JP) 2008-03-26 EP disclosed