SCHEMBL470984

SCHEMBL470984

CCOC(=O)c1cc2nc(Cl)c(NNC(=O)CC3CC3)nc2cc1CC

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 4/20 0.36
TDP1 Q9NUW8 1/20 0.36
P2RX7 Q99572 3/20 0.35
TP53 P04637 1/20 0.35
GRM1 Q13255 2/20 0.34
MELK Q14680 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HIF1A Q16665 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
OPRK1 P41145 1/20 0.33
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15374852 0.92 ALDH1A1 (0.38) P2RX7TP53GRM1POLBMAPT
SCHEMBL12060112 0.85 ALDH1A1 (0.38) P2RX7POLBMAPTALDH1A1KDM4E
SCHEMBL470985 0.82 ALDH1A1 (0.39) P2RX7GRM1POLBGAAMAPT
SCHEMBL15374840 0.76 GAA (0.40) GRM1POLBGAAALDH1A1KDM4E
SCHEMBL15374842 0.69 PGK1 (0.42) GAAKDM4E
SCHEMBL10053817 0.69 GAA (0.39) POLBGAAALDH1A1KDM4ELMNA
SCHEMBL471042 0.69 KDM4E (0.43) GRM1GAAMAPTALDH1A1L3MBTL1
SCHEMBL12060039 0.67 IDH1 (0.34) POLBGAAALDH1A1KDM4EOPRK1
SCHEMBL12043375 0.65 ALDH1A1 (0.41) P2RX7TP53POLBGAAMAPT
SCHEMBL10053819 0.65 GAA (0.42) P2RX7TP53POLBGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033101-A1 QUINOXALINE COMPOUND アステラス製薬株式会社 (JP) 2012-03-15 WO disclosed