SCHEMBL4710074

SCHEMBL4710074

COc1cc(Oc2ccnc3ccc(F)cc23)ccc1C(C(N)=O)c1cn[nH]c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.46
AXL P30530 5/20 0.46
PDGFRB P09619 3/20 0.46
CSF1R P07333 1/20 0.46
PDGFRA P16234 9/20 0.45
KIT P10721 2/20 0.45
FGFR2 P21802 1/20 0.45
MET P08581 4/20 0.43
MERTK Q12866 2/20 0.42
DDR2 Q16832 2/20 0.42
AURKA O14965 1/20 0.42
RIPK2 O43353 1/20 0.42
ABCB11 O95342 1/20 0.42
ABL1 P00519 1/20 0.42
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
NTRK1 P04629 1/20 0.42
LCK P06239 1/20 0.42
PGR P06401 1/20 0.42
LYN P07948 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5009415 0.89 AXL (0.45) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL4708410 0.87 KDR (0.51) KDRPDGFRBCSF1RPDGFRAMET
SCHEMBL2175230 0.78 KDR (0.53) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL2175628 0.74 MET (0.50) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL4710076 0.73 PDGFRB (0.72) KDRPDGFRBCSF1RPDGFRAFLT3
SCHEMBL2176270 0.71 PDGFRB (0.66) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL5009418 0.70 KDR (0.56) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL2173726 0.68 KDR (0.73) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL2172121 0.68 PDGFRB (0.71) KDRAXLPDGFRBCSF1RPDGFRA
SCHEMBL4514154 0.68 KDR (0.52) KDRAXLPDGFRBCSF1RPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994025-A1 QUINOLINE DERIVATIVES AstraZeneca AB (SE) 2008-11-26 EP claimed
WO-2007099326-A1 QUINOLINE DERIVATIVES ASTRAZENECA AB (SE) 2007-09-07 WO claimed
EP-1994025-A1 QUINOLINE DERIVATIVES AstraZeneca AB (SE) 2008-11-26 EP disclosed
WO-2007099326-A1 QUINOLINE DERIVATIVES ASTRAZENECA AB (SE) 2007-09-07 WO disclosed