SCHEMBL4713741

SCHEMBL4713741

N#CCCc1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NR3C2 P08235 1/20 0.43
PTPN7 P35236 6/20 0.40
DUSP3 P51452 6/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
AR P10275 2/20 0.40
VNN1 O95497 1/20 0.38
EPHX1 P07099 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KIF11 P52732 2/20 0.36
DAO P14920 1/20 0.35
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623982 0.82 PTPN7 (0.42) NR3C2PTPN7DUSP3CTSSCTSK
SCHEMBL29492591 0.82 PTPN7 (0.42) NR3C2PTPN7DUSP3CTSSCTSK
SCHEMBL4715187 0.80 MEN1 (0.57) MEN1KMT2ADAO
SCHEMBL3244152 0.78 TAAR1 (0.53) NR3C2PTPN7DUSP3ARCYP2D6
SCHEMBL2600223 0.77 CTSS (0.46) NR3C2PTPN7DUSP3CTSSCTSK
SCHEMBL27789311 0.77 NR3C2 (0.46) NR3C2PTPN7DUSP3AREPHX1
Hydrochloric Acid SCHEMBL3230959 0.77 TAAR1 (0.52) NR3C2PTPN7DUSP3ARCYP2D6
SCHEMBL3637053 0.77 NR3C2 (0.49) NR3C2PTPN7DUSP3AREPHX1
SCHEMBL10662203 0.75 PTPN7 (0.47) NR3C2PTPN7DUSP3AREPHX1
SCHEMBL9103643 0.75 MEN1 (0.52) MEN1KMT2ACYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337517-B1 PYRIMIDINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 2008-11-26 EP disclosed