SCHEMBL4713850

SCHEMBL4713850

Cc1cc(=O)c(C(=O)c2cccs2)c(C)[nH]1.Cc1cc(Cl)c(C(=O)c2cccs2)c(C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.40
ALDH1A1 P00352 4/20 0.36
ADORA1 P30542 3/20 0.36
MAPT P10636 3/20 0.36
PSMD14 O00487 1/20 0.36
MMP2 P08253 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
BRAF P15056 1/20 0.35
EP300 Q09472 1/20 0.35
KAT2A Q92830 1/20 0.35
KAT2B Q92831 1/20 0.35
HPGD P15428 1/20 0.35
KDM4E B2RXH2 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ADORA2A P29274 2/20 0.34
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3170295 0.86 ALDH1A1 (0.46) HDAC6ALDH1A1ADORA1MAPTPSMD14
SCHEMBL3186815 0.85 ADORA1 (0.47) HDAC6ALDH1A1ADORA1MAPTPSMD14
SCHEMBL4711599 0.81 NPC1 (0.40) HDAC6ALDH1A1MAPTHSD17B10NPC1
SCHEMBL4715159 0.79 HDAC6 (0.35) HDAC6ALDH1A1ADORA1MAPTPSMD14
SCHEMBL3179472 0.72 ADORA1 (0.43) ALDH1A1ADORA1MAPTPSMD14MMP2
SCHEMBL3187071 0.71 ADORA1 (0.43) HDAC6ALDH1A1ADORA1MAPTPSMD14
SCHEMBL3183945 0.67 HTT (0.50) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL3192305 0.66 NPSR1 (0.46) ALDH1A1MAPTHSD17B10NPC1RAB9A
SCHEMBL3175489 0.65 ALDH1A1 (0.43) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL3169957 0.64 ALDH1A1 (0.48) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996588-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS Torrent Pharmaceuticals Ltd (IN) 2008-12-03 EP disclosed
WO-2007100295-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS TORRENT PHARMACEUTICALS LTD (IN) 2007-09-07 WO disclosed