SCHEMBL4711599

SCHEMBL4711599

Cc1cc(=O)c(C(=O)c2ccc(Cl)cc2)c(C)[nH]1.Cc1cc(Cl)c(C(=O)c2ccc(Cl)cc2)c(C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 3/20 0.35
LMNA P02545 2/20 0.35
GAA P10253 1/20 0.35
CHEK2 O96017 1/20 0.35
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3192305 0.86 NPSR1 (0.46) NPC1RAB9AMAPK1NPSR1CYP1A2
SCHEMBL3179849 0.84 ALDH1A1 (0.46) NPC1RAB9AHDAC3HDAC1HDAC2
SCHEMBL4713850 0.81 HDAC6 (0.40) NPC1RAB9AHDAC6MAPK1NPSR1
SCHEMBL3169957 0.76 ALDH1A1 (0.48) NPC1RAB9AMAPK1CYP1A2CYP3A4
SCHEMBL13531552 0.74 ALDH1A1 (0.50) NPC1RAB9AMAPK1NPSR1ALDH1A1
SCHEMBL3183945 0.73 HTT (0.50) NPC1RAB9AMAPK1NPSR1ALDH1A1
SCHEMBL3175489 0.72 ALDH1A1 (0.43) NPC1RAB9ACYP1A2ALDH1A1HPGD
SCHEMBL10392166 0.68 RAB9A (0.56) NPC1RAB9AHDAC1HDAC6MAPK1
SCHEMBL900419 0.65 ALDH1A1 (0.58) NPC1RAB9AMAPK1ALDH1A1HPGD
SCHEMBL6652987 0.65 KMT2A (0.45) NPC1RAB9AMAPK1NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996588-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS Torrent Pharmaceuticals Ltd (IN) 2008-12-03 EP disclosed
WO-2007100295-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS TORRENT PHARMACEUTICALS LTD (IN) 2007-09-07 WO disclosed