SCHEMBL4714713

SCHEMBL4714713

CCN(C1CCNC1)S(=O)(=O)c1ccc2[nH]c(=O)c3[nH]ccc3c2c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.55
SLC6A4 P31645 12/20 0.55
KCNH2 Q12809 5/20 0.45
RXFP1 Q9HBX9 1/20 0.43
SLC6A3 Q01959 7/20 0.38
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP2D6 P10635 3/20 0.34
PARG Q86W56 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butyric Acid SCHEMBL4166193 0.92 SLC6A2 (0.48) SLC6A2SLC6A4KCNH2RXFP1SLC6A3
Butyric Acid SCHEMBL4157864 0.92 SLC6A2 (0.48) SLC6A2SLC6A4KCNH2RXFP1SLC6A3
SCHEMBL4717249 0.83 MAPT (0.44) SLC6A2SLC6A4KCNH2RXFP1SLC6A3
SCHEMBL3247263 0.81 SLC6A2 (0.49) SLC6A2SLC6A4KCNH2RXFP1HTT
SCHEMBL3247259 0.81 SLC6A2 (0.49) SLC6A2SLC6A4KCNH2RXFP1HTT
Butyric Acid SCHEMBL4159473 0.79 RXFP1 (0.40) SLC6A2SLC6A4KCNH2RXFP1SLC6A3
SCHEMBL4717207 0.78 MAPT (0.47) SLC6A2SLC6A4RXFP1PARGKDM4E
Butyric Acid SCHEMBL4159661 0.78 RXFP1 (0.38) SLC6A2RXFP1HTTTDP1KDM4E
Butyric Acid SCHEMBL4161016 0.78 RXFP1 (0.38) SLC6A2RXFP1HTTTDP1KDM4E
SCHEMBL4717707 0.78 RXFP1 (0.40) RXFP1PARGKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2008-03-19 EP claimed
WO-2007003611-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2007-01-11 WO claimed