SCHEMBL4714980

SCHEMBL4714980

CCOC(=O)CC(=O)c1cc(F)c(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 2/20 0.42
MGLL Q99685 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
MGAM O43451 1/20 0.41
SI P14410 1/20 0.41
MGAM2 Q2M2H8 1/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
MIF P14174 1/20 0.40
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1241168 0.92 GAA (0.49) TDP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL30680417 0.91 ALDH1A1 (0.42) TDP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL30181504 0.88 MEN1 (0.42) TDP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL29007819 0.88 MEN1 (0.42) TDP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL7009795 0.87 TDP1 (0.41) TDP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL6217850 0.86 KDM4E (0.51) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL8875853 0.86 GAA (0.48) MEN1KMT2AGAACYP1A2CYP2C19
SCHEMBL29943543 0.84 GAA (0.47) MEN1KMT2AGAACYP1A2CYP2C19
SCHEMBL28816302 0.84 GAA (0.47) MEN1KMT2AALDH1A1GAACYP1A2
SCHEMBL8183324 0.84 MEN1 (0.44) TDP1MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5077429-A 7-AMINO-1-CYCLOPROPYL-4-OXO-1,4-DIHYDRO-QUINOLINE- AND NAPHTHYRIDINE-3-CARBOXYLIC ACIDS, PROCESSES FOR THEIR PREPARATION AND ANTIBACTERIAL AGENTS CONTAINING THESE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1991-12-31 US claimed
CN-119264049-A Norfloxacin Star synthesizing method 中南大学 2025-01-07 CN disclosed
CN-116693375-B Synthesis method of 2, 4-dichloro-5-fluoro acetophenone 山东国邦药业有限公司 2023-11-24 CN disclosed
CN-116693375-A Synthesis method of 2, 4-dichloro-5-fluoro acetophenone 山东国邦药业有限公司 2023-09-05 CN disclosed
CN-116462631-A Synthetic method of norfloxacin 青海夏都医药有限公司 2023-07-21 CN disclosed
CN-115650831-B Synthetic method of 2, 4-dichloro-5-fluoro acetophenone 山东国邦药业有限公司 2023-03-28 CN disclosed
CN-115650831-A Synthetic method of 2, 4-dichloro-5-fluoro acetophenone 山东国邦药业有限公司 2023-01-31 CN disclosed
CN-109422726-B Blocking agent of CD47/SIRP alpha and application thereof 华东理工大学 2022-10-28 CN disclosed
CN-108440291-B Method for dehydrogenation and self-coupling of 1, 3-dicarbonyl compound under catalysis of visible light 南京工业大学 2020-08-28 CN disclosed
US-20140073631-A1 ANTIVIRAL AND ANTIMICROBIAL COMPOUNDS VYMED CORPORATION (US) 2014-03-13 US disclosed
EP-0230053-A2 7-(Substituted)piperazinyl-1-ethyl-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids AMERICAN CYANAMID COMPANY (US) 1987-07-29 EP disclosed
US-4670444-A 7-amino-1-cyclopropyl-4-oxo-1, 4-dihydro-quinoline-and naphthyridine-3-carboxylic acids and antibacterial agents containing these compounds BAYER AKTIENGESELLSCHAFT (DE) 1987-06-02 US disclosed
US-4620007-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1986-10-28 US disclosed
US-4611080-A Preparation of halogenated aroylacetic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1986-09-09 US disclosed
US-4563448-A PHYTOPATHOGENS BAYER AKTIENGESELLSCHAFT (DE) 1986-01-07 US disclosed
US-4563459-A FUNGICIDES AND BACTERICIDES FOR AGRICULTURAL USE BAYER AKTIENGESELLSCHAFT (DE) 1986-01-07 US disclosed
US-4559341-A Quinolonecarboxylic acids and antibacterial agents containing these compounds BAYER AKTIENGESELLSCHAFT (DE) 1985-12-17 US disclosed
US-4559342-A Quinolone acids and antibacterial agents containing these compounds BAYER AKTIENGESELLSCHAFT (DE) 1985-12-17 US disclosed
US-4547503-A 1-Cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-[4-(oxo-alkyl)-1-piperazinyl]quinoline-3-carboxylic acids and their derivatives, and antibacterial agents containing them BAYER AKTIENGESELLSCHAFT (DE) 1985-10-15 US disclosed
US-4544658-A FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 1985-10-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140073631-A1 ANTIVIRAL AND ANTIMICROBIAL COMPOUNDS GDA, GMPS, GANC TDP1 337/4885MEN1 4700/4885KMT2A 4199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.