SCHEMBL4715221

SCHEMBL4715221

O=C(O)c1cc2c(ccc(=O)n2-c2ccc3[nH]ccc3c2)n1Cc1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 14/20 0.51
CCR9 P51686 1/20 0.41
GPR35 Q9HC97 1/20 0.38
TNIK Q9UKE5 1/20 0.37
BRD4 O60885 1/20 0.37
MCHR1 Q99705 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4711667 0.92 KDM4E (0.41) CCR2TNIKBRD4MCHR1MAPT
SCHEMBL4716301 0.89 MAPT (0.44) CCR2TNIKBRD4MAPT
SCHEMBL5119050 0.83 CCR2 (0.62) CCR2CCR9GPR35MAPT
SCHEMBL4715116 0.82 CCR2 (0.55) CCR2CCR9GPR35BRD4MAPT
SCHEMBL4715213 0.76 CCR2 (0.51) CCR2BRD4MAPT
SCHEMBL4711188 0.74 BRD4 (0.53) CCR2BRD4MAPT
SCHEMBL4717022 0.74 CCR2 (0.49) CCR2BRD4MAPT
SCHEMBL4712174 0.74 MAPT (0.51) CCR2BRD4MAPT
SCHEMBL4715522 0.73 RGS4 (0.48) CCR2BRD4MAPT
SCHEMBL4715185 0.73 BRD4 (0.48) CCR2BRD4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7456286-B2 Bicyclic heteroaromatic compounds as kinase inhibitors UCB PHARMA, S.A. (BE) 2008-11-25 US disclosed
EP-1549648-B1 BICYCLIC HETEROAROMATIC COMPOUNDS AS KINASE INHIBITORS UCB PHARMA SA (BE) 2008-11-12 EP disclosed
US-20060122212-A1 Bicyclic heteroaromatic compounds as kinase inhibitors CELLTECH R&D LIMITED (GB) 2006-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060122212-A1 Bicyclic heteroaromatic compounds as kinase inhibitors MAP2K2, MAP2K7, MAP2K3 CCR2 333/4885CCR9 901/4885GPR35 2404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.