SCHEMBL4717573

SCHEMBL4717573

O=[C]NCCCc1ccc2[nH]cnc2n1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 1/20 0.36
CDK2 P24941 1/20 0.31
CTSA P10619 2/20 0.31
ALDH1A1 P00352 1/20 0.31
KDM4E B2RXH2 1/20 0.31
XDH P47989 2/20 0.31
MAPK14 Q16539 1/20 0.31
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23554436 0.70 ALDH1A1 (0.41) POLA1CDK2CTSAALDH1A1KDM4E
SCHEMBL1998243 0.68 ALDH1A1 (0.37) POLA1CDK2CTSAALDH1A1KDM4E
SCHEMBL4718044 0.67 MTNR1A (0.34)
SCHEMBL4718040 0.66 CYP2C9 (0.45)
SCHEMBL5255150 0.65 HRH3 (0.51) ALDH1A1LMNAHSD17B10
SCHEMBL19629639 0.65 KDM4E (0.37) POLA1CDK2CTSAALDH1A1KDM4E
SCHEMBL18937619 0.65 ALDH1A1 (0.37) POLA1CDK2CTSAALDH1A1KDM4E
SCHEMBL8479069 0.64 ITGAV (0.57)
SCHEMBL2008297 0.63 ALDH1A1 (0.44) CDK2CTSAALDH1A1KDM4EMAPK14
SCHEMBL2188616 0.62 CTNNB1 (0.47) CDK2CTSAALDH1A1KDM4EMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed