SCHEMBL4718674

SCHEMBL4718674

COc1cc(OC)cc(-c2nn(-c3cc(N4CCC(N(C)C)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
FGFR2 P21802 1/20 0.36
MCHR1 Q99705 4/20 0.35
FLT3 P36888 1/20 0.35
HTR1B P28222 1/20 0.35
UGCG Q16739 1/20 0.34
NOTUM Q6P988 1/20 0.34
PLK1 P53350 1/20 0.34
SOS1 Q07889 2/20 0.34
KCNH2 Q12809 1/20 0.34
F10 P00742 2/20 0.33
F2 P00734 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724584 0.92 ITGB2 (0.40) PDE4APDE4BPDE4CPDE4DMCHR1
SCHEMBL4722544 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4722323 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724510 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724513 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719501 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724695 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719498 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719376 0.89 NOTUM (0.49) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4722244 0.89 AAK1 (0.37) PDE4APDE4BPDE4CPDE4DMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed