SCHEMBL4722544

SCHEMBL4722544

COc1cc(OC)cc(-c2nn(-c3cc(N4CCC(C(F)(F)F)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
UGCG Q16739 1/20 0.36
F10 P00742 7/20 0.33
F2 P00734 3/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
KCNH2 Q12809 1/20 0.33
GRM7 Q14831 1/20 0.33
HRH3 Q9Y5N1 2/20 0.32
PTGS2 P35354 1/20 0.32
NOTUM Q6P988 2/20 0.31
GAA P10253 1/20 0.31
S1PR1 P21453 1/20 0.31
ACACB O00763 1/20 0.31
SLC6A9 P48067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724510 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724695 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719498 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4724513 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4722323 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4719501 0.90 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4718674 0.90 PDE1B (0.37) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4721093 0.89 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DUGCG
SCHEMBL4722930 0.88 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DUGCG
Hydrochloric Acid SCHEMBL4719632 0.88 CHRM1 (0.36) PDE4APDE4BPDE4CPDE4DUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed