SCHEMBL4719129

SCHEMBL4719129

COc1cc(OC)cc(-c2nn(-c3cc(OCCO)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.40
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
GRM7 Q14831 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TSHR P16473 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
F10 P00742 2/20 0.32
PARP1 P09874 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718698 0.96 HRH3 (0.41) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4723575 0.93 HRH3 (0.40) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4719309 0.91 PDE4A (0.39) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4721150 0.91 PDE4A (0.42) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4719466 0.87 PDE4A (0.41) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4723846 0.86 PDE4B (0.38) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4722089 0.86 PDE4A (0.36) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4719764 0.85 PDE4A (0.41) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4720223 0.85 PDE4A (0.41) HRH3PDE4APDE4BPDE4CPDE4D
SCHEMBL4719833 0.84 PDE4A (0.35) HRH3PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed