SCHEMBL4719985

SCHEMBL4719985

O=[C]NCCCCNc1nc2ncccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.43
NUDT1 P36639 1/20 0.41
BCHE P06276 1/20 0.41
TRPC3 Q13507 1/20 0.41
TRPC4 Q9UBN4 1/20 0.41
TRPC5 Q9UL62 1/20 0.41
PDE5A O76074 1/20 0.40
DAGLA Q9Y4D2 1/20 0.39
RIPK1 Q13546 1/20 0.39
KMT2A Q03164 1/20 0.38
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
AURKB Q96GD4 1/20 0.37
HPSE Q9Y251 1/20 0.37
TSHR P16473 1/20 0.37
TP53 P04637 1/20 0.36
XDH P47989 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385517 0.81 NUDT1 (0.49) SLC2A1NUDT1BCHETRPC3TRPC4
SCHEMBL4718040 0.80 CYP2C9 (0.45) NUDT1PDE5ADAGLAKMT2AMETAP2
SCHEMBL4714905 0.80 BCHE (0.65) SLC2A1BCHETRPC3TRPC4TRPC5
SCHEMBL5399298 0.77 NUDT1 (0.44) SLC2A1NUDT1PDE5ADAGLAKMT2A
Hydrochloric Acid SCHEMBL6251675 0.76 NUDT1 (0.43) SLC2A1NUDT1PDE5ADAGLAKMT2A
SCHEMBL4714500 0.71 FAAH (0.40) DAGLA
SCHEMBL178884 0.71 SLC2A1 (0.56) SLC2A1
SCHEMBL19377809 0.71 SLC2A1 (0.52) SLC2A1TP53
SCHEMBL3997802 0.71 PDE5A (0.50) NUDT1PDE5ARIPK1KMT2AMETAP2
SCHEMBL28284325 0.71 TP53 (0.63) NUDT1PDE5ADAGLAKMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed