SCHEMBL4720045

SCHEMBL4720045

[CH]1CCCc2cccnc2N1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
TSHR P16473 1/20 0.33
NPY5R Q15761 1/20 0.31
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
CYP1A2 P05177 1/20 0.30
GRM5 P41594 1/20 0.30
IDH1 O75874 2/20 0.30
NUDT1 P36639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL325377 0.89 ADRA2A (0.36) ADRA2AADRA2BADRA2CCYP1A2IDH1
SCHEMBL450139 0.76
SCHEMBL29416448 0.75 NNMT (0.44) ADRA2AADRA2BADRA2CTSHRNPY5R
SCHEMBL38950 0.75 NNMT (0.44) ADRA2AADRA2BADRA2CTSHRNPY5R
SCHEMBL2608519 0.73 TSHR (0.41) ADRA2AADRA2BADRA2CTSHRNPY5R
Hydrochloric Acid SCHEMBL31063054 0.73 NNMT (0.42) ADRA2AADRA2BADRA2CTSHRNPY5R
Hydrochloric Acid SCHEMBL21777851 0.73 NNMT (0.42) ADRA2AADRA2BADRA2CTSHRNPY5R
SCHEMBL30903257 0.73 TSHR (0.41) ADRA2AADRA2BADRA2CTSHRNPY5R
SCHEMBL6641301 0.70 NNMT (0.38) TSHRNPY5RGRM5NUDT1
SCHEMBL29376210 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed