SCHEMBL4720152

SCHEMBL4720152

CCCOc1ccc(C(=O)OC)cc1C#N

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.64
HPGD P15428 1/20 0.64
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAOA P21397 1/20 0.43
CYP2C19 P33261 1/20 0.43
SCN1A P35498 1/20 0.43
KCNH2 Q12809 1/20 0.43
SCN2A Q99250 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SCN3A Q9NY46 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
XDH P47989 1/20 0.43
MAPT P10636 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25315154 0.89 ALDH1A1 (0.56) ALDH1A1HPGDNPC1TP53RAB9A
SCHEMBL5874030 0.89 ALDH1A1 (0.56) ALDH1A1HPGDNPC1TP53RAB9A
SCHEMBL21854424 0.88 ALDH1A1 (0.55) ALDH1A1HPGDNPC1TP53RAB9A
SCHEMBL16188294 0.86 ALDH1A1 (0.67) ALDH1A1HPGDXDHMAPT
SCHEMBL177429 0.86 ALDH1A1 (0.84) ALDH1A1HPGDXDH
SCHEMBL27195921 0.85 ALDH1A1 (0.53) ALDH1A1HPGDNPC1TP53RAB9A
SCHEMBL30863455 0.85 ALDH1A1 (0.53) ALDH1A1HPGDNPC1TP53RAB9A
SCHEMBL2564871 0.85 ALDH1A1 (0.62) ALDH1A1HPGDHSD17B10MAPT
SCHEMBL8148281 0.83 CA1 (0.52) ALDH1A1HPGDTP53HSD17B10CYP1A2
SCHEMBL13515782 0.83 HPGD (0.53) ALDH1A1HPGDNPC1TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
EP-1942899-A2 MITOTIC KINESIN INHIBITORS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
EP-1742907-A4 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2008-01-02 EP disclosed
WO-2007056056-A2 MITOTIC KINESIN INHIBITORS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed
EP-1742907-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2007-01-17 EP disclosed
WO-2005107762-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2005-11-17 WO disclosed