SCHEMBL8148281

SCHEMBL8148281

COC(=O)c1ccc(C#N)c(C#N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
CA12 O43570 2/20 0.52
CA7 P43166 2/20 0.52
CA9 Q16790 2/20 0.52
CA14 Q9ULX7 2/20 0.52
XDH P47989 1/20 0.52
MAPT P10636 5/20 0.49
ALDH1A1 P00352 5/20 0.47
USP2 O75604 1/20 0.47
HPGD P15428 3/20 0.47
KDM4E B2RXH2 3/20 0.47
GAA P10253 3/20 0.47
HSD17B10 Q99714 2/20 0.47
GLA P06280 2/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
ATM Q13315 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105391 0.91 ALDH1A1 (0.59) CA1CA2CA12CA7CA9
SCHEMBL28880690 0.87 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL8007448 0.87 RAB9A (0.49) CA1CA2CA12CA7CA9
SCHEMBL3717515 0.86 ERN1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL1807138 0.86 XDH (0.54) XDHMAPTLMNA
SCHEMBL30488306 0.86 XDH (0.54) XDHMAPTLMNA
SCHEMBL5874030 0.86 ALDH1A1 (0.56) XDHMAPTALDH1A1HPGDHSD17B10
SCHEMBL536163 0.86 S1PR3 (0.51) CA1CA2CA12CA7CA9
SCHEMBL2427132 0.86 CA1 (0.62) CA1CA2CA12CA7CA9
SCHEMBL4598114 0.86 KDM4E (0.57) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2700641-A1 Azulenocyanine analogue compounds comprising anchoring group, method of making the same, and their use as dye for dye-sensitized solar cells Solvay SA (BE) 2014-02-26 EP disclosed
EP-1391451-B1 2-IMINOPYRROLIDINE DERIVATES EISAI R&D MAN CO LTD (JP) 2011-11-23 EP disclosed
EP-2385039-A1 2-Iminoisoindolinone derivatives as thrombin receptor antagonists Eisai R&D Management Co., Ltd. (JP) 2011-11-09 EP disclosed
US-7244730-B2 2-iminopyrrolidine derivatives EISAI CO., LTD (JP) 2007-07-17 US disclosed
US-7244730-B2 2-iminopyrrolidine derivatives EISAI CO., LTD (JP) 2007-07-17 US disclosed
US-6077853-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 2000-06-20 US disclosed
EP-0951285-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-10-27 EP disclosed
US-5939439-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-08-17 US disclosed
WO-1998029119-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1998-07-09 WO disclosed