SCHEMBL4720668

SCHEMBL4720668

CCOC(=O)OC1CN(C2CCN(C)CC2)CCN1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
CHRM1 P11229 2/20 0.36
TP53 P04637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
PKM P14618 1/20 0.32
MAPK1 P28482 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629209 1.00 ALDH1A1 (0.39) ALDH1A1CHRM1TP53TDP1SMN1; SMN2
SCHEMBL4719811 0.82 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2
SCHEMBL4629096 0.82 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2
SCHEMBL3311722 0.79 ALDH1A1 (0.40) ALDH1A1CHRM1TP53TDP1SMN1; SMN2
SCHEMBL1206605 0.79 ALDH1A1 (0.40) ALDH1A1CHRM1TP53TDP1SMN1; SMN2
SCHEMBL2330898 0.71 ALDH1A1 (0.43) ALDH1A1MEN1KMT2A
SCHEMBL4014963 0.71 ALDH1A1 (0.43) ALDH1A1MEN1KMT2A
SCHEMBL9330353 0.71 SCN1A (0.49) ALDH1A1CHRM1SMN1; SMN2MEN1KMT2A
SCHEMBL12881559 0.71 CHRM1 (0.51) ALDH1A1CHRM1SMN1; SMN2MEN1KMT2A
SCHEMBL2567582 0.70 SLC6A2 (0.43) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP disclosed
EP-1558600-A1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-08-03 EP disclosed
WO-2004037810-A1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-06 WO disclosed