SCHEMBL4720787

SCHEMBL4720787

COc1cc(OC)cc(-c2nn(-c3cc(N4CC[C@@H](NC(=O)C(C)C)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
F10 P00742 5/20 0.36
PDE2A O00408 1/20 0.36
ACACB O00763 1/20 0.35
UGCG Q16739 1/20 0.35
KMT2A Q03164 1/20 0.35
GLS O94925 5/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720791 1.00 MTNR1A (0.36) MTNR1AMTNR1BF10PDE2AACACB
SCHEMBL4724110 0.93 SMPD3 (0.40) MTNR1AMTNR1BF10ACACBUGCG
SCHEMBL4720535 0.93 SMPD3 (0.40) MTNR1AMTNR1BF10ACACBUGCG
SCHEMBL4720529 0.93 SMPD3 (0.40) MTNR1AMTNR1BF10ACACBUGCG
SCHEMBL4721705 0.91 MTNR1A (0.42) MTNR1AMTNR1BF10UGCGKMT2A
SCHEMBL4721701 0.91 MTNR1A (0.42) MTNR1AMTNR1BF10UGCGKMT2A
SCHEMBL4720911 0.90 MTNR1A (0.50) MTNR1AMTNR1BF10UGCGKMT2A
SCHEMBL4720913 0.90 MTNR1A (0.50) MTNR1AMTNR1BF10UGCGKMT2A
Hydrochloric Acid SCHEMBL4719632 0.89 CHRM1 (0.36) F10UGCGMCHR1
SCHEMBL4721983 0.87 NOTUM (0.40) ACACBUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed