SCHEMBL4721701

SCHEMBL4721701

CCC(=O)N[C@@H]1CCN(c2ccc(C(F)(F)F)c(-n3nc(-c4cc(OC)cc(OC)c4)c4c(c3=O)CCC4)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
F10 P00742 5/20 0.36
KMT2A Q03164 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
UGCG Q16739 1/20 0.34
CYP2C9 P11712 2/20 0.34
GRIA2 P42262 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
GAK O14976 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
RIPK1 Q13546 1/20 0.33
TTK P33981 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721705 1.00 MTNR1A (0.42) MTNR1AMTNR1BF10KMT2ACYP11B1
SCHEMBL4720911 0.94 MTNR1A (0.50) MTNR1AMTNR1BF10KMT2AUGCG
SCHEMBL4720913 0.94 MTNR1A (0.50) MTNR1AMTNR1BF10KMT2AUGCG
SCHEMBL4724110 0.92 SMPD3 (0.40) MTNR1AMTNR1BF10UGCGITGB2
SCHEMBL4720529 0.92 SMPD3 (0.40) MTNR1AMTNR1BF10UGCGITGB2
SCHEMBL4720535 0.92 SMPD3 (0.40) MTNR1AMTNR1BF10UGCGITGB2
SCHEMBL4720787 0.91 MTNR1A (0.36) MTNR1AMTNR1BF10KMT2AUGCG
SCHEMBL4720791 0.91 MTNR1A (0.36) MTNR1AMTNR1BF10KMT2AUGCG
Hydrochloric Acid SCHEMBL4719632 0.88 CHRM1 (0.36) F10UGCGHRH4
SCHEMBL4720118 0.86 SMPD3 (0.36) F10UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed