SCHEMBL4720957

SCHEMBL4720957

COc1cc(-c2nn(-c3cc(N4CCCC4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(N)=O)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
TGFBR1 P36897 3/20 0.35
ACVR1 Q04771 3/20 0.35
KCNK3 O14649 2/20 0.34
MAPT P10636 2/20 0.34
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
HTR2A P28223 2/20 0.34
PDE10A Q9Y233 1/20 0.33
C5AR1 P21730 1/20 0.33
UGCG Q16739 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720300 0.90 SMPD3 (0.35) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4720304 0.90 SMPD3 (0.35) PDE4APDE4BPDE4CPDE4DKCNK3
SCHEMBL4722298 0.90 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DTGFBR1
SCHEMBL4720459 0.89 F10 (0.40) MAPTF2F10
SCHEMBL4724946 0.87 TDP1 (0.39) MAPTF2F10ALDH1A1HPGD
SCHEMBL4724533 0.87 SMPD3 (0.46)
SCHEMBL4724531 0.87 SMPD3 (0.46)
SCHEMBL4724669 0.87 MAPT (0.35) MAPTF2F10MEN1ALDH1A1
SCHEMBL14101733 0.80 F10 (0.38) MAPTF2F10MEN1ALDH1A1
SCHEMBL4724420 0.79 P2RX7 (0.35) F2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed