SCHEMBL4722058

SCHEMBL4722058

COc1cc(OC)cc(-c2nn(-c3cc(NCCNC(=O)OC(C)(C)C)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
RAF1 P04049 1/20 0.37
BRAF P15056 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
BRD4 O60885 5/20 0.36
DRD2 P14416 4/20 0.34
SCD O00767 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
DYRK1A Q13627 1/20 0.33
AGTR1 P30556 1/20 0.33
AGTR2 P50052 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725015 0.96 BRD4 (0.38) PDE3BPDE3ADDB1CRBNRAF1
SCHEMBL4721889 0.88 SMN1; SMN2 (0.32) BRD4SCDSMN1; SMN2AGTR1AGTR2
SCHEMBL4721552 0.87 SCD (0.40) SCDSMN1; SMN2EPHX2
SCHEMBL4723445 0.87 SMN1; SMN2 (0.35) BRAFSCDSMN1; SMN2
SCHEMBL14101911 0.86 PDE4A (0.35) SCDSMN1; SMN2
SCHEMBL14101915 0.86 PDE4A (0.36) SCDSMN1; SMN2
SCHEMBL4720454 0.85 PDE4A (0.38) SCDSMN1; SMN2
SCHEMBL4765721 0.85 PDE4A (0.36) SCDSMN1; SMN2
SCHEMBL4722084 0.85 PDE4A (0.35) SCDSMN1; SMN2
SCHEMBL4721953 0.84 PDE4A (0.36) SCDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed