SCHEMBL4725015

SCHEMBL4725015

COc1cc(OC)cc(-c2nn(-c3cc(NCCCNC(=O)OC(C)(C)C)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.38
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
DYRK1A Q13627 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
DRD2 P14416 4/20 0.35
EPHX2 P34913 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721889 0.90 SMN1; SMN2 (0.32) BRD4EPHX2AGTR1AGTR2KDM4E
SCHEMBL4721552 0.89 SCD (0.40) EPHX2KDM4EKMT2A
SCHEMBL4720999 0.89 PDE4A (0.35) BRD4RAF1BRAFEPHX2AGTR1
SCHEMBL4719833 0.88 PDE4A (0.35) KDM4EKMT2A
SCHEMBL4765721 0.88 PDE4A (0.36) KDM4EKMT2A
SCHEMBL4722084 0.88 PDE4A (0.35) KDM4EKMT2A
SCHEMBL4720622 0.87 AAK1 (0.34) RAF1BRAFEPHX2KMT2A
SCHEMBL4722253 0.87 PDE4A (0.35) KDM4EKMT2A
SCHEMBL4723364 0.87 PDE4A (0.35) KDM4EKMT2A
SCHEMBL4721809 0.87 SCD (0.41) KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed