SCHEMBL4722220

SCHEMBL4722220

COc1cc(OC)cc(-c2nn(-c3cc(N4CC(CNC(C)=O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
NQO2 P16083 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
F10 P00742 3/20 0.33
PTGS2 P35354 1/20 0.33
UGCG Q16739 1/20 0.33
MAOA P21397 3/20 0.32
ACACB O00763 1/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
MAOB P27338 2/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
LMNA P02545 1/20 0.32
PTGS1 P23219 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722947 0.94 MAPT (0.39) GRIA2UGCGACACBALDH1A1MAPT
SCHEMBL4719850 0.89 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4722276 0.89 UGCG (0.36) GRIA2PDE4APDE4BPDE4CPDE4D
SCHEMBL4721342 0.88 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4721967 0.87 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DF10
SCHEMBL4719026 0.86 ACACB (0.38) GRIA2SMN1; SMN2F10PTGS2UGCG
SCHEMBL4719505 0.86 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4721533 0.85 NOTUM (0.39) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4720798 0.85 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL4721217 0.85 PDE4A (0.33) PDE4APDE4BPDE4CPDE4DSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed