SCHEMBL4722316

SCHEMBL4722316

COc1cncc(-c2nn(-c3cc(N4CCC(NC(C)=O)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CCO)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
SMPD3 Q9NY59 8/20 0.35
CCNC P24863 2/20 0.35
CDK8 P49336 2/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
DDR1 Q08345 2/20 0.33
CREBBP Q92793 2/20 0.33
F10 P00742 2/20 0.32
SUV39H2 Q9H5I1 1/20 0.32
SMPD2 O60906 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722313 1.00 ITGB2 (0.36) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4722251 0.94 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4766491 0.94 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4722374 0.94 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4724569 0.92 MTNR1A (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4724566 0.92 MTNR1A (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4719238 0.90 ABL1 (0.38) F10
SCHEMBL4719240 0.90 ABL1 (0.38) F10
SCHEMBL4721048 0.89 ITGB2 (0.38) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4721051 0.89 ITGB2 (0.38) ITGB2ICAM1ITGALSMPD3CCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed