SCHEMBL4721048

SCHEMBL4721048

COc1cncc(-c2nn(-c3cc(N4CC[C@@H](NC(C)=O)C4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.38
ICAM1 P05362 1/20 0.38
ITGAL P20701 1/20 0.38
SMPD3 Q9NY59 11/20 0.38
CCNC P24863 3/20 0.38
CDK8 P49336 3/20 0.38
SMPD2 O60906 1/20 0.36
FPR1 P21462 1/20 0.36
FPR2 P25090 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721051 1.00 ITGB2 (0.38) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4724110 0.93 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720535 0.93 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720529 0.93 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4722313 0.89 ITGB2 (0.36) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4722316 0.89 ITGB2 (0.36) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4720969 0.89 ABL1 (0.41) ITGB2ICAM1ITGALCYP11B1CYP11B2
SCHEMBL4720971 0.89 ABL1 (0.41) ITGB2ICAM1ITGALCYP11B1CYP11B2
SCHEMBL4722276 0.87 UGCG (0.36) ITGB2ICAM1ITGALSMPD3CCNC
SCHEMBL4720787 0.86 MTNR1A (0.36) CCNCCDK8MTNR1AMTNR1BACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed