SCHEMBL4722339

SCHEMBL4722339

CCN(C)c1cc(-c2cccc(OC)c2)nn(-c2ccccc2N)c1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
KLK3 P07288 1/20 0.40
BACE1 P56817 4/20 0.38
TLR8 Q9NR97 1/20 0.38
CCR2 P41597 1/20 0.38
MAOB P27338 1/20 0.36
EGFR P00533 1/20 0.36
POLB P06746 1/20 0.36
BRD4 O60885 1/20 0.35
MET P08581 1/20 0.35
RIPK2 O43353 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720679 0.90 CCR2 (0.39) HDAC1ADORA3ADORA2AADORA1KLK3
SCHEMBL14101815 0.89 CCR2 (0.38) HDAC1ADORA3ADORA2AADORA1KLK3
SCHEMBL4723051 0.89 SLC16A3 (0.42) HDAC1ADORA3ADORA2AADORA1KLK3
SCHEMBL4721280 0.88 SLC16A3 (0.45) HDAC1ADORA3ADORA2AADORA1CCR2
SCHEMBL4719664 0.88 CCR2 (0.38) HDAC1ADORA3ADORA2AADORA1KLK3
SCHEMBL4722315 0.85 ADORA3 (0.48) ADORA3ADORA2AADORA1CCR2POLB
SCHEMBL4766385 0.85 HDAC1 (0.39) HDAC1ADORA3ADORA2AADORA1CCR2
SCHEMBL4722471 0.85 ADORA3 (0.43) HDAC1ADORA3ADORA2AADORA1KLK3
SCHEMBL4722444 0.85 NPC1 (0.42) CCR2
SCHEMBL4722621 0.84 CCR2 (0.40) ADORA3ADORA2AADORA1KLK3CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed