SCHEMBL4722926

SCHEMBL4722926

COc1cc(OC)cc(-c2nn(-c3cc(N4CCC(NC(C)=O)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(N)=O)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.37
ICAM1 P05362 1/20 0.37
ITGAL P20701 1/20 0.37
SMPD3 Q9NY59 13/20 0.37
SMPD2 O60906 1/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
FPR1 P21462 1/20 0.34
FPR2 P25090 1/20 0.34
ACACB O00763 1/20 0.34
F10 P00742 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722923 1.00 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4721648 0.94 MTNR1A (0.39) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4721652 0.94 MTNR1A (0.39) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720117 0.91 SMPD3 (0.38) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720123 0.91 SMPD3 (0.38) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720195 0.91 SMPD3 (0.38) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4720193 0.91 SMPD3 (0.38) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4724531 0.91 SMPD3 (0.46) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4724533 0.91 SMPD3 (0.46) ITGB2ICAM1ITGALSMPD3SMPD2
SCHEMBL4724420 0.90 P2RX7 (0.35) ITGB2ICAM1ITGALF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed