SCHEMBL4723310

SCHEMBL4723310

COc1cc(OC)cc(-c2nn(-c3cc(N4CC[C@@H](NC(C)=O)C4)ccc3C(F)(F)F)c(=O)c3[nH]ccc23)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 3/20 0.40
ICAM1 P05362 3/20 0.40
ITGAL P20701 3/20 0.40
SMPD3 Q9NY59 10/20 0.39
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CCNC P24863 2/20 0.35
CDK8 P49336 2/20 0.35
SMPD2 O60906 1/20 0.35
FPR1 P21462 1/20 0.35
FPR2 P25090 1/20 0.35
BTK Q06187 1/20 0.35
ACACB O00763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723315 1.00 ITGB2 (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4721888 0.90 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4721614 0.90 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4721621 0.90 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4718873 0.88 P2RX7 (0.35) ITGB2ICAM1ITGAL
SCHEMBL4718877 0.88 P2RX7 (0.35) ITGB2ICAM1ITGAL
SCHEMBL4722039 0.85 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4721308 0.85 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4721312 0.85 ITGB2 (0.37) ITGB2ICAM1ITGALSMPD3MTNR1A
SCHEMBL4720535 0.85 SMPD3 (0.40) ITGB2ICAM1ITGALSMPD3MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed