SCHEMBL4723914

SCHEMBL4723914

CCOC(=O)Cc1c[nH]c2cc([N+](=O)[O-])ccc12

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.61
PTPRA P18433 1/20 0.56
PKLR P30613 1/20 0.55
CYP2C19 P33261 2/20 0.54
MAPT P10636 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
NQO2 P16083 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HTT P42858 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11554842 0.90 PKM (0.61) PKMPKLRMAPTMEN1KMT2A
SCHEMBL4260125 0.88 PKM (0.55) PKMPTPRAPKLRCYP2C19MAPT
SCHEMBL14823139 0.82 PKM (0.70) PKMCYP2C19MAPTMEN1KMT2A
SCHEMBL22777919 0.82 PTPRA (0.67) PKMPTPRAPKLRCYP2C19MAPT
SCHEMBL7380735 0.81 PTPRA (0.73) PKMPTPRAPKLRCYP2C19MAPT
SCHEMBL10265469 0.81 PKM (0.69) PKMPTPRAPKLRCYP2C19MAPT
SCHEMBL5175380 0.81 PKM (0.68) PKMCYP2C19MAPTMEN1KMT2A
SCHEMBL22777978 0.80 PTPRA (0.58) PKMPTPRAPKLRCYP2C19MAPT
SCHEMBL10289733 0.80 PKM (0.67) PKMCYP2C19MAPTMEN1KMT2A
SCHEMBL4261621 0.80 PKM (0.67) PKMCYP2C19MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1883451-A2 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY Neuraxon Inc. (CA) 2008-02-06 EP disclosed
WO-2007063418-A2 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2007-06-07 WO disclosed