SCHEMBL7380735

SCHEMBL7380735

CCOC(=O)[C@@H](N)Cc1c[nH]c2cc([N+](=O)[O-])ccc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.73
CYP2C19 P33261 1/20 0.71
SCN9A Q15858 3/20 0.52
PKM P14618 1/20 0.51
PKLR P30613 1/20 0.51
TACR1 P25103 2/20 0.51
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
NQO2 P16083 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
MPO P05164 1/20 0.43
TSHR P16473 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43
HIF1A Q16665 1/20 0.43
ITGB2 P05107 1/20 0.42
ICAM1 P05362 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288107 0.90 PTPRA (0.75) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL22288108 0.90 PTPRA (0.75) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL20931031 0.90 PTPRA (0.75) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL3519524 0.85 PTPRA (1.00) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL30789181 0.85 PTPRA (1.00) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL30381729 0.85 PTPRA (1.00) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL145392 0.85 PTPRA (1.00) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL2965137 0.85 PTPRA (1.00) PTPRACYP2C19SCN9APKMPKLR
SCHEMBL16366296 0.82 PTPRA (0.73) PTPRACYP2C19PKMPKLRMAPT
SCHEMBL22316600 0.82 PTPRA (0.73) PTPRACYP2C19PKMPKLRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010077-A Tranquilizers A/S FERROSAN (DK) 1991-04-23 US disclosed
EP-0030254-B1 BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR THERAPEUTICAL USE SCHERING AKTIENGESELLSCHAFT (DE) 1984-10-31 EP disclosed
US-4371536-A TRANQUILIZERS A/S FERROSAN (DK) 1983-02-01 US disclosed
EP-0030254-A1 Beta-carbolin-3-carboxylic acid derivatives, pharmaceutical compositions containing them and their therapeutical use SCHERING AKTIENGESELLSCHAFT (DE) 1981-06-17 EP disclosed