SCHEMBL4724313

SCHEMBL4724313

CCN(C)c1cc(-c2cccc(OC)c2)nn(-c2cc(N3CCOCC3)ccc2Br)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1B1 Q16678 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GSK3B P49841 1/20 0.41
GAK O14976 1/20 0.40
PRKDC P78527 1/20 0.40
HSD17B10 Q99714 2/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PTGS2 P35354 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721837 0.92 CYP1A2 (0.42) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4722204 0.92 CYP1A2 (0.42) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4723078 0.91 CYP1A2 (0.41) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4723982 0.91 GAA (0.51) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4723765 0.90 GAK (0.42) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4720635 0.90 MEN1 (0.42) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4724172 0.90 CYP1A2 (0.41) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4764880 0.89 PRKDC (0.43) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4719606 0.89 MEN1 (0.41) CYP1A2CYP1A1CYP1B1MEN1KMT2A
SCHEMBL4722684 0.89 MEN1 (0.43) CYP1A2CYP1A1CYP1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed