SCHEMBL4724660

SCHEMBL4724660

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(-c4cccnn4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724001 0.89 PDE4A (0.36) NOTUMPDE4APDE4BPDE4CPDE4D
SCHEMBL4719842 0.88 PDE4A (0.38) NOTUMPDE4APDE4BPDE4CPDE4D
SCHEMBL4720712 0.86
SCHEMBL4721383 0.86 BRD4 (0.32)
SCHEMBL4723242 0.85
SCHEMBL4719140 0.84
SCHEMBL4723635 0.84 PDE4A (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL4766566 0.82
SCHEMBL4719532 0.79 PDE4A (0.38) NOTUMPDE4APDE4BPDE4CPDE4D
SCHEMBL4723419 0.79 MEN1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed