SCHEMBL4723635

SCHEMBL4723635

COc1cc(C)cc(-c2nn(-c3cc(-c4cccnn4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
GRM7 Q14831 1/20 0.32
ROS1 P08922 2/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724001 0.93 PDE4A (0.36) PDE4APDE4BPDE4CPDE4D
SCHEMBL4719842 0.91 PDE4A (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL4765008 0.88 NTRK1 (0.31)
SCHEMBL4723868 0.85 BRD4 (0.31) GRM7ROS1
SCHEMBL4724660 0.84 NOTUM (0.31) PDE4APDE4BPDE4CPDE4D
SCHEMBL14101906 0.83 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4722014 0.83 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4720784 0.83 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4724951 0.83 NTRK1 (0.32) GRM7
SCHEMBL4720223 0.82 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DGRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed