SCHEMBL4721383

SCHEMBL4721383

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(-c4cccnn4)ccc3C(F)(F)F)c(=O)c3c2CC(C)N3)c1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.32
CREBBP Q92793 2/20 0.32
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720712 0.93
SCHEMBL4720286 0.90 BRD4 (0.32) BRD4CREBBPP2RX7
SCHEMBL4724660 0.86 NOTUM (0.31)
SCHEMBL4723868 0.85 BRD4 (0.31) BRD4CREBBP
SCHEMBL4721734 0.83 P2RX7 (0.31) P2RX7
SCHEMBL4719906 0.82 BRD4 (0.34) BRD4CREBBP
SCHEMBL4723242 0.81
SCHEMBL4719140 0.81
SCHEMBL4766566 0.78
SCHEMBL4721949 0.77 NTRK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed