SCHEMBL4724895

SCHEMBL4724895

CC(=O)CCc1sc2cnccc2c1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 3/20 0.52
GLA P06280 2/20 0.52
GAA P10253 2/20 0.52
HPGD P15428 1/20 0.52
CASP1 P29466 1/20 0.52
HTT P42858 1/20 0.52
CASP7 P55210 1/20 0.52
NCOA1 Q15788 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RCE1 Q9Y256 1/20 0.52
NCOA3 Q9Y6Q9 1/20 0.52
TDO2 P48775 1/20 0.36
GSK3B P49841 2/20 0.35
RPS6KA3 P51812 2/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765086 0.77 KDM4E (0.50) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL5622384 0.73 HPGD (0.64) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL15512118 0.70 KDM4E (0.68) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL7836288 0.69 KDM4E (1.00) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL4724459 0.69 KDM4E (0.70) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL4723975 0.69 KDM4E (0.73) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL8216031 0.68 AOC1 (0.52) ALDH1A1KDM4EGLAGAACDK8
SCHEMBL19587052 0.68 GAA (0.53) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL4766200 0.68 KDM4E (0.44) ALDH1A1KDM4EGLAGAAHPGD
Hydrochloric Acid SCHEMBL28051932 0.67 GAA (0.51) ALDH1A1KDM4EGLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934228-A2 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF Array Biopharma, Inc. (US) 2008-06-25 EP disclosed
WO-2007027855-A2 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2007-03-08 WO disclosed