SCHEMBL4721809

SCHEMBL4721809

COc1cc(OC)cc(-c2nn(-c3cc(NCCNC(C)=O)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCD O00767 12/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.35
F10 P00742 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
GRIA2 P42262 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718769 0.96 SCD (0.40) SCDMTNR1AMTNR1BSMN1; SMN2F10
SCHEMBL4721552 0.96 SCD (0.40) SCDMTNR1AMTNR1BSMN1; SMN2F10
SCHEMBL4722058 0.91 PDE3B (0.39) SCDSMN1; SMN2
SCHEMBL14101739 0.90 PDE4A (0.36) SCDSMN1; SMN2F10PDE4APDE4B
SCHEMBL4722089 0.90 PDE4A (0.36) SCDSMN1; SMN2F10PDE4APDE4B
SCHEMBL4723445 0.89 SMN1; SMN2 (0.35) SCDSMN1; SMN2F10PDE4APDE4B
SCHEMBL4722572 0.89 PDE4A (0.37) SCDSMN1; SMN2PDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL4720194 0.89 PDE4A (0.36) SCDSMN1; SMN2F10PDE4APDE4B
SCHEMBL4724043 0.89 F10 (0.42) SMN1; SMN2F10PDE4APDE4BPDE4C
SCHEMBL4721102 0.89 PDE4A (0.37) SCDSMN1; SMN2F10PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed