SCHEMBL4725264

SCHEMBL4725264

O=C(CN1C(=O)C2(CCNCC2)c2ccccc21)N1CCN(C2CCC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 12/20 0.49
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
OPRM1 P35372 4/20 0.45
OPRK1 P41145 1/20 0.45
GFER P55789 1/20 0.42
DDR1 Q08345 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005817 0.81 OPRL1 (0.60) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3762803 0.78 OPRL1 (0.57) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3762842 0.76 OPRL1 (0.58) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3774344 0.76 EGLN1 (0.44) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3766135 0.74 OPRL1 (0.61) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3769763 0.73 EGLN1 (0.48) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL3178584 0.73 OPRL1 (0.66) OPRL1OPRM1OPRK1
SCHEMBL3773817 0.72 EGLN1 (0.54) OPRL1OPRM1OPRK1
SCHEMBL3763129 0.72 OPRM1 (0.55) OPRL1KDM4EALDH1A1OPRM1OPRK1
SCHEMBL29444522 0.71 DDR1 (0.59) OPRL1DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909797-A2 DIPIPERAZINYL KETONES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2008-04-16 EP disclosed
WO-2007016496-A2 DIPIPERAZINYL KETONES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-02-08 WO disclosed