SCHEMBL4725463

SCHEMBL4725463

COc1cc(NCCCC(C)N)c2ncccc2c1C1CCCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
HSP90AA1 P07900 9/20 0.55
HSP90AB1 P08238 9/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
KDM4E B2RXH2 2/20 0.55
MAPT P10636 2/20 0.55
TDP2 O95551 1/20 0.55
ALDH1A1 P00352 1/20 0.55
FGB P02675 1/20 0.55
POLB P06746 1/20 0.55
GAA P10253 1/20 0.55
THRB P10828 1/20 0.55
TSHR P16473 1/20 0.55
NR4A1 P22736 1/20 0.55
HTT P42858 1/20 0.55
RECQL P46063 1/20 0.55
RAB9A P51151 1/20 0.55
BLM P54132 1/20 0.55
TDP1 Q9NUW8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6274409 0.99 MEN1 (0.55) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL6288073 0.84 MEN1 (0.43) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL6274163 0.82 MEN1 (0.62) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL5083232 0.81 KDM4E (0.57) HSP90AA1HSP90AB1KDM4EMAPTALDH1A1
SCHEMBL4727333 0.80 KDM4E (0.56) HSP90AA1HSP90AB1KDM4EMAPTALDH1A1
SCHEMBL4727652 0.74 MEN1 (0.43) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL4725352 0.74 NSD2 (0.59) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL5086649 0.73 NSD2 (0.58) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
Quinocide SCHEMBL157174 0.72 MEN1 (1.00) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2
Quinocide SCHEMBL29720457 0.72 MEN1 (1.00) MEN1KMT2AHSP90AA1HSP90AB1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021210-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-02-21 WO disclosed