Cyclopropane Carboxylic Acid

Cyclopropane Carboxylic Acid

SCHEMBL4725700

CC(=O)Nc1nc(N2CCOCC2)c2nc(-c3ccc(N)cc3)cnc2n1.O=C(O)C1CC1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.52
NEK2 P51955 4/20 0.44
PIK3CA P42336 2/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CG P48736 1/20 0.43
ATR Q13535 1/20 0.41
MTOR P42345 4/20 0.40
JAK2 O60674 1/20 0.40
MOK Q9UQ07 1/20 0.40
PIK3R1 P27986 1/20 0.40
ADK P55263 2/20 0.39
STAT3 P40763 1/20 0.39
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3761910 0.93 NOS1 (0.56) NOS1PIK3CAPIK3CDPIK3CGATR
SCHEMBL4725703 0.80 NOS1 (0.49) NOS1PIK3CAPIK3CDPIK3CGATR
SCHEMBL3770114 0.76 NOS1 (0.64) NOS1ATRJAK2ADK
SCHEMBL3766613 0.76 NOS1 (0.63) NOS1PIK3CAPIK3CDPIK3CGATR
SCHEMBL4450316 0.75 NOS1 (0.82) NOS1PIK3CAPIK3CDPIK3CGMTOR
SCHEMBL3752841 0.75 PIK3CA (0.49) NOS1PIK3CAPIK3CDPIK3CGMTOR
SCHEMBL4458075 0.73 NOS1 (0.64) NOS1PIK3CAPIK3CGATRMTOR
SCHEMBL4448737 0.72 NOS1 (0.61) NOS1ATRJAK2STAT3
SCHEMBL3770209 0.71 NOS1 (0.71) NOS1PIK3CAPIK3CGATRMTOR
SCHEMBL3769685 0.71 NOS1 (0.73) NOS1PIK3CAPIK3CGATRMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009079-A2 SUBSTITUTED PTERIDINES USEFUL FOR THE TREATMENT AND PREVENTION OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed