SCHEMBL472582

SCHEMBL472582

OC1[C@H](O)C(n2cnc3c(C4CCOC4)ncnc32)O[C@@H]1CNc1nc2ccccc2o1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.47
ADORA1 P30542 6/20 0.47
ADORA2A P29274 4/20 0.47
ADORA2B P29275 2/20 0.47
SLC29A1 Q99808 2/20 0.47
SLC28A1 O00337 1/20 0.47
TP53 P04637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PAX8 Q06710 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3276677 1.00 ADORA3 (0.47) ADORA3ADORA1ADORA2AADORA2BSLC29A1
Acetone SCHEMBL472485 0.96 ADORA1 (0.45) ADORA3ADORA1ADORA2AADORA2BSLC29A1
SCHEMBL13384997 0.86 ADORA1 (0.67) ADORA3ADORA1ADORA2AADORA2BSLC29A1
Acetone SCHEMBL472483 0.77 AHCY (0.38) ADORA3ADORA1ADORA2AADORA2BSLC29A1
Acetone SCHEMBL472736 0.76 ADORA1 (0.62) ADORA3ADORA1ADORA2AADORA2BSLC29A1
Acetone SCHEMBL472703 0.75 ADORA1 (0.52) ADORA3ADORA1ADORA2AADORA2BSLC29A1
SCHEMBL472527 0.74 ADORA1 (0.67) ADORA3ADORA1ADORA2AADORA2BSLC29A1
SCHEMBL6397659 0.74 ADORA1 (0.74) ADORA3ADORA1ADORA2AADORA2BSLC29A1
SCHEMBL13384992 0.73 ADORA1 (0.51) ADORA3ADORA1ADORA2AADORA2BSLC29A1
SCHEMBL6901588 0.67 DOT1L (0.67) ADORA3ADORA1ADORA2AADORA2BSLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2412716-A1 Partial and full agonists of A1 adenosine receptors CV THERAPEUTICS, INC. (US) 2012-02-01 EP disclosed