SCHEMBL4726334

SCHEMBL4726334

COc1ccc(-c2ccccn2)c(C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
RUNX1 Q01196 1/20 0.50
CCR1 P32246 1/20 0.47
CCR5 P51681 1/20 0.47
CCR8 P51685 1/20 0.47
FFAR1 O14842 2/20 0.47
SYK P43405 2/20 0.46
KMT2A Q03164 2/20 0.45
KDR P35968 1/20 0.45
MEN1 O00255 1/20 0.45
PKM P14618 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GRM5 P41594 1/20 0.45
HSP90AA1 P07900 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
NPY5R Q15761 1/20 0.44
TGFBR1 P36897 1/20 0.44
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780198 0.87 NPC1 (0.50) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL5379182 0.83 SYK (0.56) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL30525959 0.83 SYK (0.56) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL5326831 0.83 IDH1 (0.58) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL29496938 0.83 SYK (0.56) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL10560080 0.82 NPC1 (0.49) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL17751232 0.82 HSP90AA1 (0.52) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL17069071 0.81 CLK4 (0.53) NPC1RAB9ACCR1CCR5CCR8
SCHEMBL12946320 0.81 SYK (0.50) NPC1RAB9ARUNX1CCR1CCR5
SCHEMBL29496943 0.80 SYK (0.56) NPC1RAB9ARUNX1CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed
EP-2802594-B1 METAL COMPLEXES WITH DIBENZO[F,H]QUINOXALINES UDC IRELAND LTD (IE) 2017-04-19 EP disclosed
EP-1966343-B1 ELECTROLUMINESCENT METAL COMPLEXES WITH TRIAZOLES UDC IRELAND LTD (IE) 2017-04-19 EP disclosed
US-8680760-B2 Beta-diketone ancillary ligands and their metal complexes used in organic optoelectronic devices NATIONAL TSING HUA UNIVERSITY (TW) 2014-03-25 US disclosed
US-8017774-B2 Producing method for iridium complex CANON KABUSHIKI KAISHA (JP) 2011-09-13 US disclosed
WO-2008024953-A2 TRANSITION METAL-CATALYZED ALKYLATION OF C-H BONDS WITH ORGANOBORON REAGENTS BRANDEIS UNIVERSITY (US) 2008-02-28 WO disclosed
WO-2008024953-A2 TRANSITION METAL-CATALYZED ALKYLATION OF C-H BONDS WITH ORGANOBORON REAGENTS BRANDEIS UNIVERSITY (US) 2008-02-28 WO disclosed
US-20070232803-A1 PRODUCING METHOD FOR IRIDIUM COMPLEX CANON KABUSHIKI KAISHA (JP) 2007-10-04 US disclosed
WO-2006127948-A2 N-TERMINALLY MODIFIED GLP-1 RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-11-30 WO disclosed
WO-2004046103-A2 ARYLPYRIDINE COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2004-06-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232803-A1 PRODUCING METHOD FOR IRIDIUM COMPLEX LAGE3, EML4, INTS9 NPC1 3553/4885RAB9A 1578/4885RUNX1 1666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.