SCHEMBL4726414

SCHEMBL4726414

COc1ccc(NC(=S)NC2CCN(c3nccc4ccccc34)CC2)cc1.Cc1ccc(NC(=S)NC2CCN(c3nccc4ccccc34)CC2)cc1.S=C(Nc1ccccc1Cl)NC1CCN(c2nccc3ccccc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.51
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.44
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583157 0.89 MALT1 (0.51) MALT1ALDH1A1
SCHEMBL4583236 0.87 ALDH1A1 (0.54) MALT1ALDH1A1POLB
SCHEMBL4582726 0.87 POLB (0.53) MALT1ALDH1A1POLB
SCHEMBL4584076 0.81 PKM (0.54) MALT1ALDH1A1POLB
SCHEMBL4583601 0.80 KMT2A (0.52) MALT1ALDH1A1
SCHEMBL4725033 0.80 MALT1 (0.47) MALT1
SCHEMBL4725551 0.79 EGFR (0.43) ALDH1A1
SCHEMBL4582850 0.79 ALDH1A1 (0.53) MALT1ALDH1A1CCNE1CDK2
SCHEMBL4582822 0.79 ALDH1A1 (0.51) ALDH1A1
SCHEMBL4583335 0.78 MEN1 (0.55) MALT1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008028690-A1 1-(HET)ARYL-3-[HETARYL-PIPERIDIN-4-YL]-THIOUREAS AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-03-13 WO disclosed