SCHEMBL4726527

SCHEMBL4726527

COCCN(c1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
CYP2E1 P05181 1/20 0.34
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SYK P43405 1/20 0.31
CFTR P13569 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4726531 1.00 ALDH1A1 (0.39) ALDH1A1CYP2E1APOBEC3AAPOBEC3GOPRM1
SCHEMBL4795067 0.94 ALDH1A1 (0.38) ALDH1A1OPRM1OPRD1KDM4ELMNA
SCHEMBL4795076 0.94 ALDH1A1 (0.38) ALDH1A1OPRM1OPRD1KDM4ELMNA
SCHEMBL4794493 0.93 CYP2E1 (0.34) ALDH1A1CYP2E1APOBEC3AAPOBEC3GSYK
SCHEMBL4794496 0.93 CYP2E1 (0.34) ALDH1A1CYP2E1APOBEC3AAPOBEC3GSYK
SCHEMBL4794177 0.91 ALDH1A1 (0.37) ALDH1A1APOBEC3AAPOBEC3GOPRM1OPRD1
SCHEMBL4794178 0.91 ALDH1A1 (0.37) ALDH1A1APOBEC3AAPOBEC3GOPRM1OPRD1
SCHEMBL4838987 0.90 CYP2E1 (0.36) ALDH1A1CYP2E1APOBEC3AAPOBEC3GKDM4E
SCHEMBL4838993 0.90 CYP2E1 (0.36) ALDH1A1CYP2E1APOBEC3AAPOBEC3GKDM4E
Ammonia Solution, Strong SCHEMBL4156138 0.89 CYP2E1 (0.36) ALDH1A1CYP2E1APOBEC3AAPOBEC3GKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed